PIK293 free base · Synonyms: PIK-293 · PIK 293

PIK-293, an analog of IC87114, is a PI3K inhibitor.

For research use only. Not for human or veterinary use.

Target PI3K

Research area Metabolic Disease Cancer

Purity >98% Stock Inquire

Data Sheet SDS COA

PIK293 structure

CAS No.: 900185-01-5

Download structure (.mol)

Pack sizes & pricing

Size	Price	SKU	Stock
100 mg	USD 498.00	BP-02483-100mg	In stock	Get quote
250 mg	USD 980.00	BP-02483-250mg	In stock	Get quote
500 mg	USD 1,590.00	BP-02483-500mg	In stock	Get quote
1 g	USD 2,550.00	BP-02483-1g	In stock	Get quote
2 g	USD 4,080.00	BP-02483-2g	In stock	Get quote
3 g	USD 4,890.00	BP-02483-3g	In stock	Get quote
5 g	USD 6,520.00	BP-02483-5g	In stock	Get quote

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Description

PIK-293, an analog of IC87114, is a PI3K inhibitor, with IC50 values of 0.24 μM, 10 μM, 25 μM and 100 μM for p110δ, p110β, p110γ and p110α, respectively .

Identifiers

SMILES: CC1=CC=CC=C1N1C(=O)C2=C(C=CC=C2C)N=C1CN1N=CC2=C(N)N=CN=C12
InChIKey: KQDBVHKNIYROHU-UHFFFAOYSA-N

Specifications

MW (average): 397.4326
Formula: C₂₂H₁₉N₇O
CAS No.: 900185-01-5
Physical state: Solid
Color: White to off-white
Shipping: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -20°C, 1 month;

Solubility

Soluble in DMSO

Documents

References

[1].Knight ZA, et al. A pharmacological map of the PI3-K family defines a role for p110alpha in insulin signaling. Cell. 2006 May 19;125(4):733-47.

Same target

Search PI3K

Same research area

Search Metabolic Disease