CDC801 free base · Synonyms: CDC-801 · CDC 801

CDC801 is a potent and orally active phosphodiesterase 4 and tumor necrosis factor-α inhibitor.

For research use only. Not for human or veterinary use.

Target Phosphodiesterase (PDE) TNF Receptor

Research area Cancer

Purity >98% Stock Inquire

Data Sheet SDS COA

CDC801 structure

CAS No.: 192819-27-5

Download structure (.mol)

Pack sizes & pricing

Size	Price	SKU	Stock
25 mg	USD 465.00	BP-01949-25mg	In stock	Get quote
50 mg	USD 665.00	BP-01949-50mg	In stock	Get quote
100 mg	USD 965.00	BP-01949-100mg	In stock	Get quote
250 mg	USD 1,465.00	BP-01949-250mg	In stock	Get quote
500 mg	Inquire	BP-01949-500mg	In stock	Inquire
1 g	Inquire	BP-01949-1g	Inquire	Inquire

Need another size or custom synthesis? Request a quote.

Description

CDC801 is a potent and orally active phosphodiesterase 4 (PDE4) and tumor necrosis factor-α (TNF-α) inhibitor with IC50 of 1.1 μM and 2.5 μM, respectively.

Biological activity

The more detailed information refer to the Compound 6b in the reference 1 (PMID:19256507)

Identifiers

SMILES: O=C(CC(N1C(C2=C(C1=O)C=CC=C2)=O)C3=CC=C(C(OC4CCCC4)=C3)OC)N
InChIKey: DDYUBCCTNHWSQM-UHFFFAOYSA-N

Specifications

MW (average): 408.4471
Formula: C₂₃H₂₄N₂O₅
CAS No.: 192819-27-5
Physical state: Solid
Color: white to off-white
Shipping: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -20°C, 1 month

Solubility

Soluble in DMSO

Documents

References

[1]. Man HW, et al. Discovery of (S)-N-[2-[1-(3-ethoxy-4-methoxyphenyl)-2-methanesulfonylethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl] acetamide (apremilast), a potent and orally active phosphodiesterase 4and tumor necrosis factor-alpha inhibitor. J Med Chem.

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