BiochemProbe — Life Science Research Reagents

Clobutinol free base

Clobutinol is a compound that has anti-tussive effects.

For research use only. Not for human or veterinary use.

Purity >98% Stock Inquire

Clobutinol structure

CAS No.: 14860-49-2

Download structure (.mol)

Pack sizes & pricing

Size Price SKU Stock
No pack sizes listed. Request a quote.

Description

Clobutinol is a compound that has anti-tussive effects. Clobutinol affects heart rate and blood pressure, it can be used for cough related research.

Biological activity

In Vitro Clobutinol (10 μM) significantly inhibits the voltage-gated outward current in hERG-expressing cells[1]. Clobutinol (0-1000 μM) inhibits the outward current in hERG transfected cells with an IC50 value of 1.9 μM In Vivo Clobutinol (1-20 mg/kg; i.v. once) has no obvious effect on the airway of guinea-pigs. Clobutinol (1 and 10 mg/kg; i.v. once) affects heart rate and mean blood pressure of guinea pigs

Identifiers

SMILES
ClC1=CC=C(C=C1)CC(O)(C)C(C)CN(C)C
InChIKey
KVHHQGIIZCJATJ-UHFFFAOYSA-N

Specifications

MW (average)
255.7840
Formula
C14H22ClNO
CAS No.
14860-49-2
Physical state
Solid
Color
White to off-white
Shipping
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.

References

[1]. Deisemann H, et al. Effects of common antitussive drugs on the hERG potassium channel current. J Cardiovasc Pharmacol. 2008 Dec;52(6):494-9.
[2]. Salonen RO. Comparison of the effects of two opioid antitussives, vadocaine hydrochloride, clobutinol and lidocaine on lung mechanics in guinea-pigs. Arzneimittelforschung. 1988 Apr;38(4A):609-12.
[3]. Takahara A, Set al. Clobutinol delays ventricular repolarization in the guinea pig heart: comparison with cardiac effects of HERG K+ channel inhibitor E-4031. J Cardiovasc Pharmacol. 2009 Dec;54(6):552-9.

Same research area

Search Cardiovascular Disease