PF-06372222 free base · Synonyms: GPCR modulator-1

GPCR modulator-1 is a negative allosteric modulator of GLP receptor.

For research use only. Not for human or veterinary use.

Target GCGR

Research area Metabolic Disease

Purity >98% Stock Inquire

Data Sheet SDS COA

PF-06372222 structure

CAS No.: 1407592-99-7

Download structure (.mol)

Pack sizes & pricing

Size	Price	SKU	Stock
10 mg	USD 498.00	BP-01885-10mg	In stock	Get quote
25 mg	USD 912.00	BP-01885-25mg	In stock	Get quote
50 mg	USD 1,396.00	BP-01885-50mg	In stock	Get quote
100 mg	USD 2,148.00	BP-01885-100mg	In stock	Get quote
500 mg	Inquire	BP-01885-500mg	In stock	Inquire
1 g	Inquire	BP-01885-1g	Inquire	Inquire

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Description

GPCR modulator-1 is a negative allosteric modulator of GLP receptor. GPCR modulator-1 has the potential for type 2 diabetes research.

Identifiers

SMILES: CC1(CC(C1)[C@H](C2=CC=C(C=C2)C(=O)NCCC(=O)O)NC3=CN=C(C=C3)N4C=C(N=C4)C(F)(F)F)C
InChIKey: MYZIDYJMNWEJMC-QHCPKHFHSA-N

Specifications

MW (average): 515.5274
Formula: C₂₆H₂₈F₃N₅O₃
CAS No.: 1407592-99-7
Physical state: Solid
Color: White to off-white
Shipping: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage: Powder 4℃, 2 years; In solvent -20℃ 1 month;

Documents

References

[1]. Gaojie Song, et al. Human GLP-1 receptor transmembrane domain structure in complex with allosteric modulators. Nature. 2017 Jun 8;546(7657):312-315.

Same research area

Search Metabolic Disease