Deucrictibant free base · Synonyms: PHA-022121

Deucrictibant is a novel and potent bradykinin receptor antagonist.

For research use only. Not for human or veterinary use.

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Data Sheet SDS COA

Deucrictibant structure

CAS No.: 2340111-58-0

Download structure (.mol)

Pack sizes & pricing

Size	Price	SKU	Stock
5 mg	USD 785.00	BP-02001-5mg	In stock	Get quote
10 mg	USD 1,085.00	BP-02001-10mg	In stock	Get quote
25 mg	USD 1,585.00	BP-02001-25mg	In stock	Get quote
50 mg	USD 2,140.00	BP-02001-50mg	In stock	Get quote
100 mg	USD 2,885.00	BP-02001-100mg	In stock	Get quote
1 g	Inquire	BP-02001-1g	In stock	Inquire

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Description

Deucrictibant (PHA-022121) is a novel and potent bradykinin receptor antagonist. PHA-022121 is a small molecule antagonist of the bradykinin B2 receptor. It has a subnanomolar affinity and is a surmountable and reversible antagonist.

Identifiers

SMILES: [2H][C@](C)(C1=C(C(=CC(=C1)F)Cl)COC2=CC=CC3=C(C=C(N=C32)C)C4=NC=NN4C)NC(=O)COC(F)F
InChIKey: ZTCLCSCHTACERP-WTDRUJNCSA-N

Specifications

MW (average): 534.9360
Formula: C₂₅H₂₃ClF₃N₅O₃
CAS No.: 2340111-58-0
Physical state: Solid
Color: White to off-white
Shipping: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage: Powder -20℃, sealed storage, away from moisture and light, 3 years; In solvent -20℃ 1 month;

Solubility

Soluble in DMSO

Documents

References

[1]. https://www.sciencedirect.com/science/article/pii/S1567576922000078

[2]. https://www.frontiersin.org/journals/pharmacology/articles/10.3389/fphar.2020.00916/full

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