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TAK-653 free base · Synonyms: TAK 653 · TAK653

TAK-653 is an AMPA receptor potentiator with minimal agonistic activity.

For research use only. Not for human or veterinary use.

Research area Neurological Disease
Purity >98% Stock Inquire

TAK-653 structure

CAS No.: 1358751-06-0

Download structure (.mol)

Pack sizes & pricing

Size Price SKU Stock
250 mg USD 550.00 BP-01876-250mg In stock Get quote
500 mg USD 750.00 BP-01876-500mg In stock Get quote
1 g USD 1,350.00 BP-01876-1g In stock Get quote
5 g Inquire BP-01876-5g Inquire Inquire

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Description

TAK-653 is an AMPA receptor potentiator with minimal agonistic activity.

Biological activity

TAK-653, an AMPA receptor potentiator with minimal agonistic activity, produces an antidepressant-like effect with a favorable safety profile in rats. In Vivo Osavampator (0.03-0.3 mg/kg, p.o., single dose) enhances visual learning and memory in normal rats. Osavampator (0.3 mg/kg, p.o., single dose) enhances sustained attention in the poor performing rats. Osavampator (0.06 mg/kg, p.o., single dose) improves working memory in monkeys. Osavampator (1 mg/kg, p.o., single dose) produces antidepressant-like effects in the rat RSBM (reduction of submissive behavior model).

Identifiers

SMILES
O=S1(N=C2C(C3=CC=C(C=C3)OC4CCCCC4)=NC(C)=CN2CC1)=O
InChIKey
PXJBHEHFVQVDDS-UHFFFAOYSA-N

Specifications

MW (average)
373.4690
Formula
C19H23N3O3S
CAS No.
1358751-06-0
Physical state
Solid
Color
White to yellow
Shipping
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage
Powder 4°C, sealed storage, away from moisture and light; In solvent -20℃ 1 month;

Solubility

Soluble in DMSO ≥ 12.5 mg/mL

References

[1]. Hara H, et al. TAK-653, an AMPA receptor potentiator with minimal agonistic activity, produces an antidepressant-like effect with a favorable safety profile in rats. Pharmacol Biochem Behav. 2021 Dec;211:173289.
[2]. Suzuki A, et al. Strictly regulated agonist-dependent activation of AMPA-R is the key characteristic of TAK-653 for robust synaptic responses and cognitive improvement [J]. Scientific Reports, 2021, 11(1): 14532.
[3]. Hara H, et al. TAK-653, an AMPA receptor potentiator with minimal agonistic activity, produces an antidepressant-like effect with a favorable safety profile in rats. Pharmacol Biochem Behav. 2021 Dec;211:173289.

Same target

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Same research area

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