Troriluzole free base
Troriluzole, a third-generation, tripeptide proagent of Riluzole , is an orally active glutamate modulator.
For research use only. Not for human or veterinary use.
Troriluzole structure
CAS No.: 1926203-09-9
Pack sizes & pricing
| Size | Price | SKU | Stock | |
|---|---|---|---|---|
| 10 mg | USD 365.00 | BP-02418-10mg | In stock | Get quote |
| 25 mg | USD 730.00 | BP-02418-25mg | In stock | Get quote |
| 50 mg | USD 1,170.00 | BP-02418-50mg | In stock | Get quote |
| 100 mg | USD 1,870.00 | BP-02418-100mg | In stock | Get quote |
| 250 mg | USD 3,740.00 | BP-02418-250mg | In stock | Get quote |
| 500 mg | Inquire | BP-02418-500mg | In stock | Inquire |
| 1 g | Inquire | BP-02418-1g | In stock | Inquire |
Need another size or custom synthesis? Request a quote.
Description
Troriluzole, a third-generation, tripeptide proagent of Riluzole , is an orally active glutamate modulator. Troriluzole reduces synaptic glutamate level and increases the synaptic glutamate absorption. Troriluzole has the potential for Alzheimer disease and generalized anxiety disorder (GAD) .
Biological activity
In Vitro Troriluzole is absorbed systemically and cleaves into riluzole by aminopeptidases.
Identifiers
- SMILES
-
O=C(CN(C)C(CNC(CN)=O)=O)NC1=NC2=CC=C(OC(F)(F)F)C=C2S1 - InChIKey
-
YBZSGIWIPOUSHY-UHFFFAOYSA-N
Specifications
- MW (average)
- 419.3790
- Formula
- C15H16F3N5O4S
- CAS No.
- 1926203-09-9
- Physical state
- Solid
- Color
- White to off-white
- Shipping
- Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
- Storage
- Powder -20°C, 3 years , 4°C, 2 years ; In solvent -20°C, 1 month
Solubility
Soluble in DMSO : 50 mg/mL